Part I: Protein Conjugates
1. Site-Specific Labeling of Proteins for Single-Molecule FRET Measurements Using Genetically Encoded Ketone Functionalities
Edward A. Lemke
2. Enzymatically-Catalyzed Conjugation of a Biodegradable Polymer to Proteins and Small Molecules Using Microbial Transglutaminase
Ahmed Besheer, Thomas C. Hertel, Jörg Kressler, Karsten Mäder, and Markus Pietzsch
3. Synthesis of Drug/Dye-Incorporated Polymer-Protein Hybrids
Sukanta Dolai, Wei Shi, Bikash Mondal, and Krishnaswami Raja
4. Dye/DNA Conjugates as Multiple Labels for Antibodies in Sensitive Fluorescence Immunoassays
Qin Zhang, Shengchao Zhu, and Liang-Hong Guo
5. Chemoselective Modification of Viral Proteins Bearing Metabolically Introduced 'Clickable' Amino Acids and Sugars
Partha S. Banerjee and Isaac S. Carrico
6. Preparation of Peptide and Other Biomolecular Conjugates through Chemoselective Ligations
Mathieu Galibert, Olivier Renaudet, Didier Boturyn, and Pascal Dumy
7. New Fluorescent Substrates of Microbial Transglutaminase and Its Application to Peptide Tag-Directed Covalent Protein Labeling
Noriho Kamiya and Hiroki Abe
8. Covalent Conjugation of Poly(Ethylene Glycol) to Proteins and Peptides: Strategies And Methods
Anna Mero, Chiara Clementi, Francesco M. Veronese, and Gianfranco Pasut
9. Extending the Scope of Site-Specific Cysteine Bioconjugation by Appending a Prelabeled Cysteine Tag to Proteins Using Protein Trans-Splicing
Tulika Dhar, Thomas Kurpiers, and Henning D. Mootz
Part II: Nucleic Acid Conjugates
10. Polyethylenimine Bioconjugates for Imaging and DNA Delivery In Vivo
Andrea Masotti and Francesco Pampaloni
11. Synthesis of a Glycomimetic Oligonucleotide Conjugate By 1,3-Dipolar Cycloaddition
Gwladys Pourceau, Albert Meyer, Jean-Jacques Vasseur, and François Morvan
12. Site-Specific DNA Labeling by Staudinger Ligation
Samuel H. Weisbrod, Anna Baccaro, and Andreas Marx
13. Improved Cellular Uptake of Antisense Peptide Nucleic Acids (PNAs) by Conjugation to a Cell-Penetrating Peptide and a Lipid Domain
Takehiko Shiraishi and Peter E. Nielsen
14. Synthesis of Oligonucleotide-Peptide Conjugates for Biomedical and Technological Applications
Anna Aviñó, Santiago Grijalvo, Sónia Pérez-Rentero, Alejandra Garibotti, Montserrat Terrazas, and Ramon Eritja
15. Amphiphilic DNA Block Copolymers: Nucleic Acid-Polymer Hybrid Materials for Diagnostics and Biomedicine
Jan Zimmermann, Minseok Kwak, Andrew J. Musser, and Andreas Herrmann
Part III: Glycosyl and Lipid Conjugates
16. Chemically Selective Liposome Surface Glyco-Functionalization
Hailong Zhang, Yong Ma, and Xue-Long Sun
17. Bioconjugation Using Mutant Glycosyltransferases for the Site-Specific Labeling of Biomolecules with Sugars Carrying Chemical Handles
Boopathy Ramakrishnan, Elizabeth Boeggeman, Marta Pasek, and Pradman K. Qasba
18. Lipid-Core-Peptide System for Self-Adjuvanting Synthetic Vaccine Delivery
Mariusz Skwarczynski and Istvan Toth
19. Coupling Carbohydrates to Proteins for Glycoconjugate Vaccine Development Using a Pentenoyl Group as a Co
